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SRT-3109

  Cat. No.:  DC26142   Featured
Chemical Structure
1204707-71-0
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More than 5000 active chemicals with high quality for research!
Field of application
SRT3109 is an antagonist of CXCR2, with a pIC50 of 8.2, and used in the research of chemokine mediated diseases.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1204707-71-0
Synonyms: SRT-3109,SRT 3109,SRT3109
SMILES: FC1=C(F)C=CC=C1CSC2=NC(NS(=O)(N3CCC3)=O)=CC(N[C@@H]([C@@H](O)CO)C)=N2
Formula: C18H23F2N5O4S2
M.Wt: 475.53
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks4°C in DMSO,6 months-80°C in DMSO
Description: SRT3109 is an antagonist of CXCR2, with a pIC50 of 8.2, and used in the research of chemokine mediated diseases.
Target: CXCR2:8.2 (pIC50)
In Vitro: SRT3109 (Example 1) is an antagonist of CXCR2, with a pIC50 of 8.2, and used in the research of chemokine mediated diseases[1].
References: [1]. Premji Meghani, et al. Pyrimidyl sulfonaminde derivative and its use for the treatment of chemokine mediated diseases. WO2010007427A1
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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