Novel inhibitors

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Cat. No.	Product Name	Field of Application
DC11765	GRK2-IN-115h hydrochloride	A highly potent and selective GRK2 inhibitor with IC50 of 18 nM. More description
DC21604	SA-57	A highly potent and selective dual FAAH/MAGL inhibitor with IC50 of 1-3 nM against FAAH, inhibits mouse (IC50=410 nM) and human (IC50=1.4 uM) MAGL. More description
DC23477	MRS-2500 tetraammonium	A highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. More description
DC23476	MRS-2500	A highly potent and selective antagonist of the platelet P2Y1 receptor with Ki of 0.78 nM. More description
DC22523	3-Deazaneplanocin A hydrochloride	A highly potent and competitive S-adenosylhomocysteine hydrolase inhibitor with Ki of 0.05 nM, also inhibits histone methyltransferase EZH2. More description
DC21592	ML165	A high-affinity, selective platelet integrin αIIbβ3 receptor antagonist with IC50 of 96 nM. More description
DC23268	MIV 150	A high-affinity, allosteric HIV-1 and HIV-2 reverse transcriptase inhibitor (NNRTI) with EC50 of 1 nM. More description
DC23757	MLS-000532223	A high affinity, selective inhibitor of Rho family GTPases with EC50 of 16-120 uM. More description
DC22860	Saframycin A	A heterocyclic quinone antibiotic that inhibits RNA synthesis in vivo and in vitro. More description
DC11564	CDK9-PROTAC	A heterobifunctional small molecule PROTAC capable of cereblon mediated proteasomal degradation of CDK9. More description
DC25080	6-Maleimidohexanoic acid N-hydroxysuccinimide ester	A heterobifunctional cross-linking reagent incorporating an extended spacer with amine and sulfhydryl reactivity. More description
DC24171	Furilazole	A herbicide safener for gramineous crops.. More description
DC23983	Pyraclonil	A herbicide agent. . More description
DC22359	Valproic acid	A HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. More description
DC22358	Valproic acid sodium salt	A HDAC inhibitor that selectively inhibits the catalytic activity of class I HDACs, and induces proteasomal degradation of HDAC2. More description
DC21845	Carbenoxolone disodium	A glycyrrhetinic acid derivative that inhibits 11β-hydroxysteroid dehydrogenase (11β-HSD), a gap junction blocker and mineralocorticoid agonist.. More description
DC21844	Carbenoxolone	A glycyrrhetinic acid derivative that inhibits 11β-hydroxysteroid dehydrogenase (11β-HSD), a gap junction blocker and mineralocorticoid agonist.. More description
DC21363	Lucerastat	A galactose analogue that is an UDP-glucose ceramide glucosyltransferase (UGCG/GCS) inhibitor (IC50=41.4 uM). More description
DC20497	PGRMC2-IN-25	A gain-of-function ligand for PGRMC2 (progesterone receptor membrane component 2) to promote adipogenesis. More description
DC21669	SNAP 5114	A GABA transport inhibitor with IC50 of 5, 21, 388 and 140 uM for hGAT-3, rGAT-2, hGAT-1 and BGT-1, respectively. More description
DC24161	Acamprosate calcium	A GABA receptor agonist and modulator of glutamatergic systems. More description
DC23737	Azaphilone-9	A fungal natural product that binds to HuR and inhibits HuR-RNA interaction in vitro with IC50 of 1.2 uM. More description
DC11489	6-alkynyl Fucose	A fucose analog that inhibits Dll-induced Notch signaling by reducing Notch ligand Dll1-Notch1 binding, but not Jag1. More description
DC22353	Gatifloxacin	A fourth-generation fluoroquinolone antibiotic that inhibits the bacterial DNA gyrase and topoisomerase IV. More description
DC22351	Gatifloxacin mesylate	A fourth-generation fluoroquinolone antibiotic that inhibits the bacterial DNA gyrase and topoisomerase IV. More description
DC22352	Gatifloxacin hydrochloride	A fourth-generation fluoroquinolone antibiotic that inhibits the bacterial DNA gyrase and topoisomerase IV. More description
DC22520	Porcine dynorphin A(1-13)	A form of dynorphin and an endogenous opioid peptide with the amino acid sequence: Tyr-Gly-Gly-Phe-Leu-Arg-Arg-Ile-Arg-Pro-Lys-Leu-Lys.. More description
DC11531	Teslexivir	A first-in-class, small molecule protein-protein inhibitor of the interaction between the E1 and E2 proteins of HPV types 6 and 11. More description
DC11707	MDVN-1003	A first-in-class, selective, orally bioavailable, dual inhibitor of BTK and PI3Kδ kinases with IC50 of 32.3 nM and 16.9 nM, respectively. More description
DC11814	cis CM-414	A first-in-class, dual inhibitor of PDE5 and HDAC that inhibits HDAC1/2/3/6 (IC50=310/490/322/91 nM, respectively) and PDE5 (IC50=60 nM). More description

Novel inhibitors

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