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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC39093 | JH-RE-06 |
JH-RE-06 is a potent REV1-REV7 interface inhibitor with an IC50 of 0.78 μM and Kd value of 0.42 μM, disrupting REV1-POL ζ-mediated mutagenic translesion synthesis (TLS).
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| DC39087 | GCN2iB |
GCN2iB is an ATP-competitive serine/threonine-protein kinase general control nonderepressible 2 (GCN2) inhibitor with IC50 of 2.4 nM.
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| DC39086 | Epertinib hydrochloride |
Epertinib hydrochloride (S-222611 hydrochloride) is a potent, orally active, reversible, and selective tyrosine kinase inhibitor of EGFR, HER2 and HER4 with IC50 of 1.48 nM, 7.15 nM and 2.49 nM, respectively. Epertinib hydrochloride (S-222611 hydrochloride) exhibits antitumor activity.
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| DC39081 | BCH |
BCH (LAT1-IN-1) is a selective and competitive inhibitor of system L amino acid transporter 1 (LAT1). BCH (LAT1-IN-1) induces apoptosis in cancer cells.
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| DC39080 | 1-Aminobenzotriazole |
1-Aminobenzotriazole (ABT, 3-Aminobenzotriazole, 1-Benzotriazolylamine, NSC 114498, NSC 656987) is a nonselective and irreversible inhibitor of cytochrome P450 (CYP) enzymes. 1-Aminobenzotriazole is also a substrate and inhibitor of N-acetyltransferase (NAT).
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| DC33598 | GSK-805 Featured |
GSK805, also known as ROR gamma-t-IN-1, is a potent, orally bioavailable retinoid-related orphan receptor gamma t (RORγt) inverse agonist that interacts with the receptor's putative ligand binding domain without exerting significant effects on DNA binding.
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| DC39055 | BIIB068 Featured |
BIIB068 is a potent, selective, reversible and orally active BTK inhibitor. BIIB068 demonstrated good kinome selectivity with good overall drug-like properties for oral dosing, was well tolerated across preclinical species at pharmacologically relevant doses with good ADME properties, and achieved >90% inhibition of BTK phosphorylation (pBTK) in humans.
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| DC9474 | Nelfinavir (Mesylate) |
Nelfinavir(AG-1341) is a potent and orally bioavailable human immunodeficiency virus HIV-1 protease inhibitor (Ki=2 nM) and is widely prescribed in combination with HIV reverse transcriptase inhibitors for the treatment of HIV infection.
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| DC25028 | AUDA Featured |
A potent inhibitor of sEH (soluble epoxide hydrolase) with IC50 of 18 nM and 69 nM for mouse sEH and human sEH, respectively.
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| DC23149 | Oseltamivir acid |
Oseltamivir acid (GS 4071, Ro 64-0802, Oseltamivir carboxylate) is a potent inhibitor of influenza neuraminidase (NA) with Ki of <1 nM for both A and B strains,showed potent activity against COVID-19(SARS-COV-2).
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| DC39019 | Y-1 Featured |
Compound Y-1 exerts the best inhibition activity (IC50
= 0.21 μM) against NA, which is better than oseltamivir
carboxylate (OSC) (IC50 = 3.04 μM) and lead AN-329/
10738021 (IC50 = 1.92 μM).
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| DC22089 | Rimeporide (EMD-87580) |
Rimeporide (EMD87580) is a potent, selective sodium hydrogen exchanger NHE1 inhibitor, show promise as potential therapeutic agents for the treatment of heart failure..
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| DC39013 | (R)-Viloxazine Hydrochloride Featured |
The (S)-isomer of Viloxazine.
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| DC39012 | (S)-Viloxazine Hydrochloride Featured |
The (S)-isomer of Viloxazine.
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| DC37997 | Leucyltyrosine |
Leucyltyrosine is a peptide.
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| DC37860 | Small cardioactive peptide A |
Small cardioactive peptide A is a neuropeptide that modulates neuromuscular synapsis in Aplysia. It also functions as neural cotransmitter in molluscs and exert a role in both the central and peripheral modulation of the control of feeding behavior.
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| DC37850 | Tetralysine |
Tetralysine is a cationic moietie that may be used in the construction of gene delivery vectors and DNA nanoparticles.
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| DC37816 | S-Adenosyl-L-homocysteine |
S-Adenosylhomocysteine is an amino acid derivative used in several metabolic pathways in most organisms. It is an intermediate in the synthesis of cysteine and adenosine.
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| DC37806 | L-Saccharopine |
L-Saccharopine is a product of breakdown of essential amino acid Lysine. Saccharopine is also part of the α-aminoadipate pathway of fungal lysine biosynthesis.
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| DC37791 | KKI 5 |
KKI 5 is a serine protease inhibitor that inhibits kallikrein and plasmin. KKI 5 may exhibit anticancer chemotherapeutic benefit and may also be used as a treatment for angioedema. In various cancer cell lines, KKI 5 alters membrane potential and increases intracellular Ca2+, inhibiting cell proliferation.
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| DC37755 | Carvyl propioate |
Carvyl propioate is a Skin / Eye Irritant.
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| DC37723 | Pidolic acid |
Pidolic acid is a cyclized derivative of L-GLUTAMIC ACID. Elevated blood levels may be associated with problems of GLUTAMINE or GLUTATHIONE metabolism.
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| DC37359 | Dichlofenthion |
Dichlofenthion is a phosphorothioate which is primarily used as a pesticide and nematicide.
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| DC37263 | 4-Hydroxymetanilic acid |
4-Hydroxymetanilic acid is a biochemical.
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| DC37111 | 4-Chlorobenzenesulfonamide |
4-Chlorobenzenesulfonamide is a sulfonamide derivative.
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| DC37087 | p-tert-Butylphenol |
p- tert- Butylphenol is a chemical compound from the group of phenols .
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| DC36832 | (+)-Gallocatechin |
(+)-Gallocatechin is a polyphenol and flavonoid that has been isolated from the leaves of tea plants and has diverse biological activities.
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| DC36802 | Lymecycline |
Lymecycline is a semisynthetic antibiotic related to TETRACYCLINE.
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| DC36748 | Benoxacor |
Benoxacor is an inert agricultural chemical that acts as an herbicide safener to protect crops from herbicide toxicity.
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| DC36550 | Dicloran |
Dicloran is a biochemical.
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