Novel specific PAK4 inhibitor, effectively inhibiting the invasion of SGC7901 cells without cytotoxicity, regulating the PAK4/LIMK1/cofilin and PAK4/SCG10 signaling pathways

Novel potent and selective binder of small subunit B of the serine palmitoyltransferase complex (SPTSSB)

Novel potent serine palmitoyl transferase (SPT) inhibitor

Novel SPOP inhibitor, suppressing the viability and inhibiting the colony formation of ccRCC cell lines driven by cytoplasmic SPOP

Pivotal intercellular signal transmitter

USP7 inhibitor from the marine sponge Stylissa massa

Novel isosteric charge-deficient spermine analogue

Novel potent sPLA2 inhibitor, selectively targeting hGIIA and hGIID

Sterol Biosynthesis Inhibitor, Fungicide

Novel p53 Stabilizer for Brain Cell Differentiation

Novel selective orally bioavailable inhibitor of p300/CBP histone acetyltransferase

Novel gamma-secretase modulator

Antibiotic, binding to the bacterial 30S ribosomal subunit, interfering with the initiation of protein synthesis and with proper protein elongation and leading to bacterial cell death

Novel anti-tuberculosis agent against intracellular Mycobacterium tuberculosis

Novel photo-controllable hydrogen sulfide donor applicable in live cells

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Novel telomerase inhibitor

Novel Programmed Death Ligand 1 (PD-L1) Binding Peptide (a Peptide Ligand for PD-L1)

Sorting inhibitor, blocking Vps16 function, one protein in the class C tethering complex, and increasing aflatoxin synthesis and export

Novel partial inhibitor of amphetamine-induced dopamine release

DAT modulator, being unique in affecting substrate uptake without impacting efflux

Human norepinephrine transporter blocker

Natural inhibitor of the Kv1.3 channels in a concentration-dependent manner

Inhibitor of constitutive and inducible STAT3 activation through the activation of SHP-2 tyrosine phosphatase

Natural analgesic, antipyretic, anti-inflammatory, and anti-tumor agent

A2A adenosine receptor agonist

Novel, selective and orally bioavailable c-Met inhibitor, exhibiting antitumor activity both in vitro and in vivo

Novel potent and selective allosteric modulator of sigma-1 receptor

Unique somatostatin receptor subtypes 2-, 4- and 5-selective analogue, effectively reducing GH secretion in human GH-secreting pituitary adenomas even in Octreotide non-responsive tumours.

Novel long-acting, reversible albumin-binding growth hormone (GH) derivative for treatment of growth hormone dificiency