Brevicornin is a flavonol from Epimedium brevicornum.

Isorhamnetin 7-O-α-L-rhamnoside shows binding affinity with COVID-19 virus main protease.

Hemiphroside B is found in Lagotis integra.

Isohericerin is an isoindolinone natural product.

Eugenol rutinoside is found in dendropanax dentiger.

Boeravinone A is found in Boerhavia diffusa L.

Ilexsaponin B3 has significant hypocholesterolemic activity.

cyclo(Phe-Ala-Gly-Arg-Arg-Arg-Gly-AEEAc) provides an avenue for developing a nonhormonal male contraceptive by blocking of GRTH/DDX25 phosphorylation.

BCECF-AM is a cell membrane permeable compound widely used as a fluorescent indicator for intracellular pH.

Aβ Fibrillization modulator 1 stabilizes Aβ monomers.

Calmodulin antagonist-1 (W-7) is a calmodulin (CaM) antagonist. Calmodulin antagonist-1 inhibits calmodulin-activated Ca2+-phosphodiesterase (PDE) (IC50=28 μM). Calmodulin antagonist-1 also inhibits trypsin-treated Ca2+-PDE (IC50=375 μM) in a competitive fashion with respect to cyclic GMP and the Ki value is 300 μM.

Compound 48/80 (Poly-p-methoxyphenethylmethylamine) is widely used in animal and tissue models as a "selective" mast cell activator. Compound 48/80 acts at the mast cell membrane to stimulate trimeric G-proteins and induces degranulation via phospholipase C and D pathways.

Idroxioleic acid ((R)-2-Hydroxyoleic acid; (R)-2-OHOA), the R enantiomer of (Rac)-Idroxioleic acid, is an orally active fatty acid that modulates the lipid composition and structure of the membranes. Idroxioleic acid has antitumor activities.

D-threo-PPMP is a potent inhibitor of glucosylceramide (GlcCer) synthase. D-threo-PPMP can block karyokinesis and reduce cyst production.

ERGi-USU-6 (mesylate) is an ERGi-USU-6 salt derivative that is a new selective inhibitor of ERG positive prostate cancer ( IC50 = 0.089 μM).

gTPA2-OMe is a potential hole transport layer candidate for perovskite solar cells (PSCs).

Antiviral agent 6 shows excellent anti-TSWV activity in vivo, and the EC50 value is 188 mg/L.

Anti-ToCV agent 1 can be used as a potential anti-ToCV drug.

Antiviral agent 7 is a peptide-based coating that can kill viruses.

APJ receptor agonist 3 is a potent and orally active APJ receptor agonist with an EC50 value of 0.027 nM.

Cyclopropenone probe 1 can specifically and efficiently modify a triple-negative breast cancer driver, glutathione S-transferase pi-1 (GSTP1), by covalently binding at the catalytic active site.

FTO-IN-4 is a potent and selective inhibitor of fat mass obesity-associated protein (FTO).

FTO-IN-5 is a potent and selective inhibitor of fat mass obesity-associated protein (FTO).

hTrkA-IN-2 is a selective hTrkA allosteric inhibitor with an IC50 value of 3.9 nM.

Antitumor agent-29 is a novel hepatocyte-targeting antitumor prodrug, which exhibits good antitumor activity and low toxic side effects.

DN-F01 has a strong inhibitory calcium-dependent effect on cardiac myofibrillar ATPase activity with an IC50 value of 11 ± 4 nmol/L.

Epyrifenacil is a newly developed herbicide.

Galectin-8-IN-1 is a selective ligand for the galectin-8 N-terminal domain (galectin-8N), with a Kd of 48 μM and 15-fold selectivity over galectin-3 and even better selectivity over the other mammalian galectins.

GT-055 (LCB18-055) is a novel broad-spectrum β-lactamase inhibitor.

CASK-IN-1 is a highly potent and selective CASK inhibitor with a Kd value of 0.022 μM.