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[D-Trp11]-Neurotensin

  Cat. No.:  DC42313  
Chemical Structure
73634-68-1
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Field of application
[D-Trp11]-Neurotensin, an analogue of Neurotensin (NT), is a selective antagonist of NT in perfused rat hearts but behaves as a full agonist in guinea pig atria and rat stomach strips. [D-Trp11]-Neurotensin can inhibit NT-induced hypotension.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 73634-68-1
Chemical Name: [D-Trp11]-Neurotensin
Synonyms: {Pyr}-LYENKPRRP-{D-Trp}-IL
Formula: C80H122N22O19
M.Wt: 1695.96
Sotrage: Please store the product under the recommended conditions in the Certificate of Analysis.
MSDS
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MSDS_25920_DC42313_73634-68-1
COA
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Cat. No. Product name Field of application
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DC44146 SORT-PGRN interaction inhibitor 1 SORT-PGRN interaction inhibitor 1 is a potent inhibitor of the sortilin-progranulin interaction with an IC50 of 2 μM.
DC42313 [D-Trp11]-Neurotensin [D-Trp11]-Neurotensin, an analogue of Neurotensin (NT), is a selective antagonist of NT in perfused rat hearts but behaves as a full agonist in guinea pig atria and rat stomach strips. [D-Trp11]-Neurotensin can inhibit NT-induced hypotension.
DC42046 [Lys8, Lys9]-Neurotensin (8-13) [Lys8, Lys9]-Neurotensin (8-13) (JMV438), a Neurotensin analog, exerts its analgesic effects through activation of the G protein-coupled receptors NTS1 and NTS2, with Ki values of 0.33 nM and 0.95 nM for hNTS1 and hNTS2 receptors, respectively.
DC41694 JMV 449 JMV 449 is a potent neurotensin receptor agonist. JMV 449 shows an IC50 of 0.5 nM in binding to mouse brain membranes and an EC50 of 1.9 nM in contracting the guinea-pig ileum. JMV 449 has highly potent and long-lasting hypothermic and analgesic effects in the mouse.
DC28455 NTRC-824 NTRC-824 (Compound 5) is a potent, selective and neurotensin-like nonpeptide neurotensin receptor type 2 (NTS2) antagonist with an IC50 of 38 nM and a Ki of 202 nM. NTRC-824 is >150-fold selectivity for NTS2 over NTS1 (Ki >30 μM).
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