VX-150|CAS 1793080-72-4|DC Chemicals

Cas No.:	1793080-72-4
Chemical Name:	(4-(2-(4-Fluoro-2-methylphenoxy)-4-(trifluoromethyl)benzamido)-2-oxopyridin-1(2H)-yl)methyl dihydrogen phosphate
Synonyms:	BDBM186573;US9163042, VX-150;VX150 VX 150;EOS-62073;EOS62073;EOS 62073
SMILES:	P(=O)(O[H])(O[H])OC([H])([H])N1C([H])=C([H])C(=C([H])C1=O)N([H])C(C1C([H])=C([H])C(C(F)(F)F)=C([H])C=1OC1C([H])=C([H])C(=C([H])C=1C([H])([H])[H])F)=O
Formula:	C₂₁H₁₇F₄N₂O₇P
M.Wt:	516.3363
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:	VX-150 is an orally active, highly selective NaV1.8 inhibitor. VX-150 has the potential for various pain indications research[1].
In Vitro:	VX-150 is an orally bioavailable pro-drug that rapidly converts into its active moiety, which is a highly selective inhibitor of NaV1.8 relative to the other sodium channel subtypes (>400-fold)[1].

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