Inhibitor of Beta_amyloid>amyloid β-mediated cellular toxicity

Novel STING Agonist

Novel, active, and less toxic anti-tuberculosis (anti-TB) agent

Novel pro-angiogenic agent, potently promoting proliferation, migration, invasion and tube formation of human umbilical vein VECs (HUVECs) in vitro

Highly selective and relatively potent group II metabotropic glutamate receptor agonist

Novel double photocaged cathepsin B activity-based probe for monitoring the light-activation by the blue fluorescence of 7-diethylamino-4-hydroxymethyl-coumarin (DEACM) and simultaneously probe the activity of cathepsin B through the green fluorescence of

Novel inhibitor of soluble epoxide hydrolase (sEH), showing good solubility, microsomal stability, and selectivity for sEH

Novel inhibitor of thioredoxin reductase (TrxR)

Antiatherosclerotic, antihyperlipidemic, antiinflammatory, antifungal, antiviral and antineoplastic

Inhibitor of the Cdc42-PBD interaction, blocking the association of Cdc42 with the PBD

Potent human sex hormone binding globulin (SHBG) ligand

Potent and selective JNK inhibitor; Analogue of SP600125 with improved potency and selectivity

Non-hydrolyzable ATP analog, acting as an effective and selective NTPDase2 inhibitor

Novel potent natural STAT3 signaling inhibitor from Polygonum cuspidatum, inhibiting cell growth and inducing apoptosis of HCC cells and HCC Cancer stem cells.

Endogenous superagonist of transient receptor potential melastatin 2 (TRPM2)

Inhibitor of cellular glycosylation; Analytical standard

Site BI- selective synergistic activator of PKA I

Lipid mediator, regulates neuronal apoptosis in traumatic brain injury (TBI)

Metabotropic Glutamate Receptor 5-selective Negative Allosteric Modulator

Novel potent activator of both human and mouse TLR4-NF-κB reporter cells and primary cells, inducing serum anti-HA and anti-NA IgG1 levels

Novel GPR88 Agonist

Novel selective inhibitor of EGFR kinase, leading to inactivation of PI3K/AKT/mTOR and Ras-Raf-MEK-ERK signal pathways

Novel Selective LXRβ Agonist

Oxysterol agonist of the liver X receptor

Novel Versatile Probe for Interrogating Histone Benzoylation and Interactions in Living Cells

Stimulator of the central nervous system, decreasing the 5-hydroxytryptamine (5-HT) and 5-hydroxyindoleacetic acid (5-HIAA) levels in brain

Concentration- and time-dependent inhibitor of the growth of NSCLC cells inducing apoptosis

Inhibitor of SykM442A S505A ASKA- (analog-sensitive kinase alleles) mediated cellular calcium flux

Natural Inhibitor for FcεRI expression on mast cell from Verbasucum thapsus L

Novel potent antiangiogenic agent, binding to VEGFR2, significantly reducing neovascularization in both ex vivo and in vivo angiogenic assays without affecting the proliferation of endothelial cells