Specific inhibitor of the histone H3 lysine 9 demethylase KDM4 in HeLa cells.

Antipsychotic and sedative agent as a potent antagonist of H1, 5-HT2A, and alpha1-adrenergic receptors

Metabolite of nicotinamide; Specific and potent inhibitor of NNMT, increasing histone methylation at H3K4 and methylated H3K4 occupancy at gene promoters

Novel Bromodomain Binding Mimic of Lysine Acetylation

Metabolite of Trifluoperazine; Antidepressant and antipsychotic

Potent NAE-hydrolyzing acid amidase (NAAA) inhibitor

AKT Inhibitor, Enhancing Gemcitabine Activity in Pancreatic Cancer Cells

EC 3.1.1.7 (Acetylcholinesterase) inhibitor, acting as an insecticide, an acaricide, an agrochemical, and a nematicide

Potent and long-acting derivative of the hormone Trenbolone

Central sugar signal in plants, regulating sucrose use and allocation, underpinning crop growth and development

Novel TGR5 agonist, reducing glycemic and dyslipidemic cardiovascular risk in animal models of diabesity

Inhibitor of histone deacetylases

Novel Highly Selective β2-Adrenoceptor Agonist as an Oral Antiasthmatic Agent

Metabolite of Resveratrol

Metabolite of Resveratrol

Natural specific inhibitor of γ-secretase, decreasing amyloid-beta levels without influencing cleavage of Notch, showing strong growth inhibitory effects on cancer cell lines and significant anti-complement activity, also acting as a PTP1B inhibitor

Natural resveratrol trimer, acting as a protein kinase C inhibitor

Novel KGA allosteric inhibitor

Novel HuR binder, modulating HuR-RNA interactions

Potent and selective NMDA agonist

Metabolite of Resveratrol

Potent I 2 -imidazoline receptor agonist

Novel Type-I Inhibitor of TIE-2

Mitochondria-activatable luciferin (MAL-Probe)

Enhancer of the cytotoxic effect of immunotoxins (ITs) which results in increased apoptosis in different cancer cells

Novel tumour progression locus 2 (Tpl2) kinase inhibitor

Novel taxane family member, reducing the brain metastatic colonization of breast cancer cells

Novel Specific Inhibitor of Type I Collagen Production in Fibrosis

Promising amyloid reducing agent by lowering the levels of Aβ.

Inhibitor of tyrosine recombinases and Holliday junction-resolving enzymes; Antibacterial