S-Enantiomer of folcisteine, a plant growth regulator

Selective kynurenine aminotransferase 2 (KAT2) inhibitor

PET precursor for NNC112

Less active enantimer of Bambuterol

Potent and selective inhibitor of PI 3-kinase ß (PI3-Kß)

Potent beta-adrenoreceptor antagonist

Natural flavonoid from the stem bark of Bolusanthus speciosus

The First Selective Orthosteric GluK3 Antagonist

Novel potent orally available allosteric TSH receptor (TSHR) agonist

Novel σ Receptor Agonist with Neuroprotective Effect

Elongation factor P (EF-P) fuction modifier

More active enantiomer of praziquantel as potent anthelmintic

Enhancer of memory function

Selective Dopamine D3 Receptor Antagonist

More active R diastereomer of Pam2Cys, acting as a potent TLR2 agonist

Inhibitor of dopamine beta-hydroxylase

Competitive Specific Inhibitor of sphingosine kinase 2 (SK2)

R-Enantiomer of folcisteine, a plant growth regulator

Negative control for UNC6852

KB-R7943 mesylate is a potent, selective inhibitor of the reverse mode of the Na+/Ca2+ exchanger (IC50 = 0.7 mM).

An aminoglycoside antibiotic similar in structure to gentamicin B1.

1-Methoxy PMS is an electron mediator for NAD(P)H-tetrazolium salt.

N-Type calcium channel inhibitor

Novel potent and selective oxytocin receptor antagonist

Micafungin(FK463) is an echinocandin antifungal drug, Micafungin inhibits the production of beta-1,3-glucan, an essential component of fungal cell walls.

Avibactam sodium(NXL-104) is a non-β-lactam β-lactamase inhibitor antibiotic.

DS-437 is a potent, selective, dual inhibitor of PRMT5 and PRMT7 with IC50 of 6.0 uM for both, DS-437 is inactive against 29 other human protein-, DNA-, and RNA-methyltransferases.

Apilimod(STA 5326) mesylate is a potent IL-12/IL-23 inhibitor, IL-12 production in cultures of IFN-r/LPS–stimulated human PBMCs is strongly inhibited by STA-5326 with an IC50 of 10 nM.

DS18561882 is a potent and isozyme-selective MTHFD2 inhibitor with GI50 of 140 nM, which also shows good oral pharmacokinetic profile.

N-Formyl-Met-Leu-Phe, also known as fMLF, is a potent neutrophil chemoattractant and the reference agonist for the G protein-coupled N-formylpeptide receptor (FPR).