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Cat. No. Product Name Field of Application Chemical Structure
DC10572 MDK35833(Oct3/4-inducer-1) Featured
MDK35833, also known as Oct3/4-inducer-1, is a potent Oct3/4-inducer.
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DC24209 MDK7229(MD2-IN-1) Featured
MDK7229, also known as MD2-IN-1 is a MD2 (Myeloid differentiation protein 2) inhibitor.
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DC10570 MDK74978(Multi-kinase inhibitor) Featured
MDK74978, also known as Multi-kinase inhibitor I, is a Multi-kinase inhibitor. MDK74978 has CAS#778274-97-8. The last 5 digit was used in its name.
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DC10571 MDK-8582(Hnps-PLA Inhibitor) Featured
MDK-8582, also known as Hnps-PLA Inhibitor, is an nhibitor of human nonpancreatic secretory Phospholipase A (hnps-PLA).
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DC10650 MDVN1003 Featured
MDVN1003 is a potent inhibitor of BTK amd PI3K delta.
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DC8712 Deoxycorticosterone acetate Featured
Deoxycorticosterone acetate is a steroid hormone produced by the adrenal gland that possesses mineralocorticoid activity and acts as a precursor to aldosterone.
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DC8906 Indinavir Featured
Indinavir(MK-639; L735524) is a potent and specific HIV protease inhibitor that appears to have good oral bioavailability.
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DC8910 Flunarizine dihydrochloride Featured
Flunarizine is a selective calcium entry blocker.
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DC8932 TG003 Featured
TG003 is a potent and ATP-competitive Cdc2-like kinase (Clk) inhibitor with IC50 of 20 nM, 200 nM, and 15 nM for Clk1, Clk2, and Clk4, respectively. No inhibitory effect on Clk3, SRPK1, SRPK2, or PKC.
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DC8939 Tolrestat Featured
Tolrestat(AY-27773) is a potent, orally active aldose reductase inhibitor with IC50 value of 35 nM.
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DC9375 GPDA Featured
GPDA(Glycylproline p-nitroanilide tosylate) is the substarate of X-Prolyl dipeptidyl-aminopeptidase in the enzyme assay.
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DC9460 CHR-6494 Featured
CHR-6494 is a potent and selective Haspin (Haploid Germ Cell-Specific Nuclear Protein Kinase) inhibitor that blocks H3T3ph phosphorylation.
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DC9500 Cevimeline (hydrochloride hemihydrate) Featured
Cevimeline hydrochloride hemihydrate, a novel muscarinic receptor agonist, is a candidate therapeutic drug for xerostomia in Sjogren's syndrome.
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DC9569 Nefazodone (hydrochloride) Featured
Nefazodone hydrochloride is an antidepressant drug.
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DC9651 Ingenol 3-angelate Featured
Ingenol 3-Angelate is a PKC(protein kinase C)activator; anti-cancer drug and an active ingredient in Euphorbia peplus.
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DC8979 Stavudine Featured
Stavudine is a nucleoside analog that inhibits reverse transcriptase and has in vitro activity against HIV.
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DC9010 Sasapyrine Featured
Salsalate is a nonsteroidal anti-inflammatory drug (NSAID).
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DC20065 PF-06733804 Featured
Trk-IN-3 is a potent pan-Trk inhibitor in cell-based assays with IC50s of 8.4 nM, 6.2 nM and 2.2 nM for TrkA, TrkB and TrkC, respectively. Anti-hyperalgesic effect.
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DC20297 6-Hydroxy-DL-DOPA Featured
6-Hydroxy-DL-DOPA is a small-molecule that disrupts with RAD52 oligomerization, inhibits ssDNA binding by RAD52 with IC50 of 1.1 uM and by RAD52 (1 209) with IC50 of 1.6 uM.
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DC20857 Calhex-231 Featured
Calhex-231 is a potent negative allosteric modulator of CaSR that blocks calcium-mediated activation with IC50 of 0.39 uM.
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DC20945 DC_AC50 Featured
DC_AC50 (DCAC50) is a small molecule that inhibits the human copper chaperones Atox1 and CCS (Kd=6.8 and 8.2 uM), blocks copper trafficking and significantly attenuates cancer cell proliferation.
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DC21002 Edelfosine Featured
Edelfosine is a synthetic lysophospholipid analog that selectively inhibits PLC with IC50 of 9.6 uM in fibroblasts and adenocarcinoma cells.
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DC20866 CC-671 Featured
CC-671 is a potent, selective, dual TTK (Mps1)/CLK2 inhibitor with IC50 of 5/3 nM, respectively.
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DC33031 CRANAD-2 Featured
CRANAD-2 is a difluoroboron-derivatized curcumins as near-infrared probe for in vivo detection of amyloid-beta deposits. Upon interacting with Abeta aggregates, CRANAD-2 undergoes a range of changes, which include a 70-fold fluorescence intensity increase, a 90 nm blue shift (from 805 to 715 nm), and a large increase in quantum yield. Moreover, this probe also shows a high affinity for Abeta aggregates (K(d) = 38.0 nM), a reasonable log P value (log P = 3), considerable stability in serum, and a weak interaction with albumin. After intravenous injection of this probe, 19-month-old Tg2576 mice exhibited significantly higher relative signal than that of the control mice over the same period of time.
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DC33238 A286982 Featured
A286982 is an inhibitor that blocks the integrin-ligand interaction between leukocyte function-associated antigen-1 (LFA-1) and intercellular adhesion molecule-1.
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DC10328 Migalastat hydrochloride Featured
Migalastat hydrochloride (1-Deoxygalactonojirimycin hydrochloride) is a potent and competitive inhibitor of α-galactosidase A (α-Gal A) with an IC50 of 0.04 μM for human α-Gal A.
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DC9275 Mirin Featured
Mirin is a Mre11-Rad50-Nbs1 (MRN)-ATM pathway inhibitor that blocks the 3' and 5' exonuclease activity associated with Mre11.
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DC10568 Mitapivat Featured
Mitapivat is an activator of pyruvate kinase isoenzyme M2 (PKM2),
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DC34085 Epiblastin A Featured
Epiblastin A is a Casein Kinase 1 (CK1) inhibitor. Epiblastin A engages CK1 isoenzymes in cell lysate and induces efficient conversion of epiblast stem cells (EpiSCs) into embryonic stem cells (cESCs).
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DC34651 EC23 Featured
EC23 is a fluorescent, voltage, indicator, action, potentials, mammalian, neurons, perturbations, cardiac, waveform, pluripotent, stem, cell-derived, cardiomyocytes
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