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| Cat. No. | Product Name | Field of Application | Chemical Structure |
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| DC12323 | CHK1-IN-2 |
CHK1-IN-2 is a checkpoint kinase 1 (CHK1) inhibitor, with an IC50 of 6 nM
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| DC12515 | Chiglitazar |
Chiglitazar (CS-038, CS038) is a potent, dual PPARα/γ dual agonist with EC50 of 1.2, 0.08, 1.7 uM for PPARα, PPARγ and PPARδ, respectively.
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| DC20338 | Chemocoxib A |
Chemocoxib A is a highly potent, selective, cytotoxic COX-2 inhibitor with IC50 of 290 nM and 90 nM for wt mCOX-2 and R120Q COX-2 mutant respectively.
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| DC12205 | CHEMBL333994 (FK-480) |
CHEMBL333994 is a potent and orally effective Cholecystokinin A (CCK-A) antagonist, with an IC50 of 0.67 nM.
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| DC5135 | Chaetominine |
Chaetominine , an alkaloidal metabolite with a new framework, was characterized from the solid-substrate culture of Chaetomium sp.
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| DC20337 | Chaetocin |
Chaetocin is a potent, specific, SAM-competitive inhibitor of histone H3K9 methyltransferase (HMT) SU(VAR)3-9 with IC50 of 0.6 uM, no actiivty against H4 Lys20-specific HMT PRSET7 and SET7/9.
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| DC7102 | CH5132799 Featured |
CH5132799 selectively inhibits class I PI3Ks, such as PI3Kα, PI3Kβ, PI3Kδ, and PI3Kγ with IC50 values of 0.014, 0.12, 0.50, and 0.36 uM, respectively; shows less inhibition of class II PI3Ks, class III PI3ks, and mTOR.
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| DC21331 | CGS 27023A |
CGS 27023A (MMI 270) is a potent, orally active MMP inhibitor with Ki of 8-43 nM for MMP1/2/3/9.
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| DC24112 | CGS 21680 |
CGS 21680 is a specific adenosine A2A subtype receptor agonist with Ki of 27 nM.
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| DC20887 | CGP-74514A hydrochloride |
CGP-74514A hydrochloride is a potent CDK1 inhibitor with IC50 of 25 nM.
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| DC23830 | CGP-53353 |
CGP-53353 (DAPH-7) is a selective inhibitor of PKCβII with IC50 of 0.41 uM, shows weak activity on PKCβI with IC50 of 3.8 uM.
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| DC11133 | CFM-4.16 |
CFM-4.16 is a CARP-1 functional mimetic (CFM) compound bind with CARP-1, stimulates CARP-1 expression and apoptosis.
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| DC23338 | CFI-401980 |
CFI-401980 is a potent, selective, novel class TTK (Tyrosine Threonine Kinase) inhibitor with Ki of 0.8 nM, HCT116 GI50 of 13 nM.
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| DC22052 | CFI02 |
CFI02 (CFI-02) is a specific inhibitor of human cytomegalovirus (HCMV) glycoprotein B-mediated fusion with IC50 of 40 nM against laboratory adapted HCMV strain AD169.
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| DC7899 | Cevipabulin(TTI 237) |
Cevipabulin, also known as TTI-237, an antimicrotubule agent, is a small synthetic molecule of triazolopyrimidine derivative with potential antitumor activity.
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| DC10226 | Cefradine |
Cephradine is a semi-synthetic cephalosporin antibiotic.
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| DC23856 | CEP-7055 |
CEP-7055 is a potent, orally active, pan inhibitor of VEGFR, CEP-7055 is the dimethylglycine ester prodrug of CEP-5214, which inhibits human VEGFR2/KDR kinase, VEGFR1/FLT-1 kinase, and VEGFR3/FLT-4 kinase with IC50 of 18 nM, 12 nM, and 17 nM.
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| DC22796 | CEP-1347 |
CEP-1347 (KT-7515) is a potent and selective MLK inhibitor that completely rescues motoneurons and inhibits JNK1 activation with IC50 of 20 nM.
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| DC12319 | Centanafadine (EB-1020) |
Centanafadine is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.
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| DC12318 | Centanafadine hydrochloride (EB-1020 (hydrochloride)) |
Centanafadine (hydrochloride) is dual norepinephrine (NE)/dopamine (DA) transporter inhibitor, also inhibits serotonin transporter, with IC50s of 6 nM, 38 nM and 83 nM for human NE, DA and serotonin transporter , respectively.
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| DC21554 | AS 703569 |
Cenisertib (AS 703569;R763) is a novel potent, orally available inhibitor of Aurora kinases, exhibits signifficant anti-proliferative activity against a wide range of tumor cells both in vitro and in vivo (A549 EC50=9 nM).
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| DC23359 | CeMMEC2 |
CeMMEC2 is a novel potent BRD4 inhibitor with IC50 of 0.9 uM, binds to both bromodomains of BRD4, comparably to (S)-JQ1..
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| DC7569 | Z-LEHD-FMK |
Cell permeable fluoromethyl ketone (FMK)-derivatized peptides act as effective irreversible Caspase inhibitors with no cytotoxic effects and, therefore, are useful tools for studying Caspase activity.
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| DC12245 | Ceftizoxime |
Ceftizoxime is a bacterial inhibitor which acts by interfering with bacterial cell wall synthesis and inhibiting cross-linking of the peptidoglycan.
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| DC9355 | Ceftibuten (dihydrate) |
Ceftibuten dihydrate is a third-generation cephalosporin antibiotic.
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| DCAPI1033 | Cefprozil hydrate (Cefzil) |
Cefprozil hydrate (Cefzil)
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| DC8687 | Cefpirome sulfate |
Cefpirome Sulfate is a fourth generation cephalosporin antibiotic.
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| DC9356 | Cefpiramide (sodium) |
Cefpiramide sodium (SM-1652; Wy-44635) is a new Pseudomonas-active cephalosporin with a broad spectrum of antibacterial activity.
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| DC20190 | Cefoxitin |
Cefoxitin is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.
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| DCAPI1038 | Cefoselis sulfate |
Cefoselis sulfate
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