Cat. No. | Product Name | Field of Application | Chemical Structure |
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DC9128 | Ramipril |
Ramipril is an angiotensin-converting enzyme (ACE) inhibitor with IC50 of 5 nM.
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DC7828 | Ramelteon |
Ramelteon is a novel melatonin receptor agonist for human MT1 and MT2 receptors and chick forebrain melatonin receptors with Ki of 14 pM, 112 pM and 23.1 pM, respectively.
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DC6918 | Ramatroban (BAY u3405) |
Ramatroban (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
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DC9479 | Raltegravir (potassium salt) |
Raltegravir potassium salt(MK0518 potassium salt) is a potent integrase (IN) inhibitor, used to treat HIV infection.
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DC9166 | Raloxifene HCl |
RaloxifeneHcl(LY156758 Hcl) is a second generation selective estrogen receptor antagonist.
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DCAPI1577 | Raloxifene |
Raloxifene hydrochloride is a selective estrogen receptor modulator (SERM), binding to ERα and ERβ. Tissue-dependently blocks or activates estrogen-induced transcription. Exhibits estrogen agonist behavior in bone but acts as an anti-estrogen in breast an
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DC8930 | Rafoxanide |
Rafoxanide is a salicylanilide used as an antiparasitic agent.
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DC21069 | Radalbuvir |
Radalbuvir (GS-9669) is a highly optimized thumb site II nonnucleoside inhibitor of HCV NS5B polymerase with binding affinity of 1.35 nM for genotype 1b.
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DC21544 | rac Pterosin B |
rac Pterosin B is a potent and specific SIK3 signaling inhibitor that suppresses SIK3 downstream cascades by up-regulating the phosphorylation levels in the SIK3 C-terminal regulatory domain.
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DC21555 | R-999636 |
R-999636 is a small molecule inhibitor that effectively inhibits the β-catenin/Tcf4 interaction with Ki of 8.8 uM in FP assay.
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DC10995 | R916562 |
R916562 (R562) is a potent, dual Axl/VEGF-R2 inhibitor with celluar IC50 of 136 nM for Axl.
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DC2068 | R547 |
R547 is a potent and selective CDK inhibitor with Ki and IC50 of 1-3 nM and 80 nM respectively.
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DC21551 | R-360163 |
R-360163 is a small molecule inhibitor that effectively inhibits the β-catenin/Tcf4 interaction with Ki of 16 uM in FP assay.
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DC22205 | R191 |
R191 (R-191) is a potent, small molecule IRAK1/4 kinase inhibitor (IRAK4 IC50=3 nM), exhibits good selectivity against a broad panel of kinases.
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DC11138 | Guanabenz acetate |
R15A inhibitor.
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DCAPI1281 | Quinine HCl dihydrate |
Quinine HCl dihydrate
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DC8691 | Quetiapine sulfoxide dihydrochloride |
Quetiapine Sulfoxide is a metabolite of Quetiapine. Quetiapine is an atypical antipsychotic approved for the treatment of schizophrenia, bipolar disorder, and along with an antidepressant to treat major depressive disorder.
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DCAPI1284 | Quercetin dihydrate (Sophoretin) |
Quercetin dihydrate (Sophoretin)
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DC22204 | QTX125 |
QTX125 (QTX-125) is a novel potent, selective HDAC6 inhibitor, displays excellent selectivity over other HDACs.
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DC5139 | QS 11 (QS11,BML-WN117) |
QS 11 is a GTPase activating protein of ADP-ribosylation factor 1 (ARFGAP1) inhibitor.
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DC12605 | QO IIR |
QO IIR is a reversible, tight-binding inhibitor inhibitor of catechol-O-methyltransferase (COMT) with IC50 of 320 nM.
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DC11478 | QM385 |
QM385 is a highly potent small molecule SPR inhibitor,that inhibits the BH4 pathway, blocking T cell proliferation and autoimmunity.
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DC12556 | QM31 |
QM31 (SVT016426, Apaf-1 inhibitor QM31) is a cytoprotective agent that inhibits the formation of the apoptosome (IC50=7.9 uM in vitro), the caspase activation complex composed by Apaf-1, cytochrome c, dATP and caspase-9.
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DC20522 | QL-X-138 |
QL-X-138 is a selective and potent BTK/MNK dual kinase inhibitor with IC50 of 8, 107.4, and 26 nM for BTK, MNK1, and MNK2, respectively.
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DC7747 | QL-IX-55 |
QL-IX-55 is a selective ATP-competitive inhibitor of mTORC1/2 with IC50s of 50/50/10-50 nM for Human mTORC1/Yeast mTORC1/Yeast mTORC2, respectively
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DC21550 | QD 325 |
QD325 is a potent redox modulator that induces Nrf2-mediated oxidative stress and unfolded protein responses in PDAC cells (IC50=0.9 uM).
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DC21549 | QD 232 |
QD 232 is a novel quinazolinedione-based redox modulator that potently inhibits Src/FAK and STAT3 phosphorylation, decreasing pancreatic cancer cell viability and migration.
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DC11040 | QCA570 |
QCA570 is a novel, highly potent efficacious BET degrader (PROTAC).
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DC11041 | QCA276 |
QCA276 is a novel potent BET proteins inhibitor with IC50/Ki of 10/.3 nM, QCA276 is the BET ligand for PROTAC QCA570.
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DC21548 | QC-6352 |
QC-6352 is a potent and selective KDM4 family inhibitor with IC50 of 104, 56, 35, and 104 nM for KDM4A, KDM4B, KDM4C, and KDM4D, respectively.
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