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BMS-P5

  Cat. No.:  DC39626   Featured
Chemical Structure
1550371-22-6
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Field of application
BMS-P5 is a Novel Peptidylarginine Deiminase 4 (PAD4) Inhibitor with pIC50 values in the range of 5-​7.5. BMS-P5 Blocks Formation of Neutrophil Extracellular Traps and Delays Progression of Multiple Myeloma. Administration of BMS-P5 to multiple myeloma-be
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1550371-22-6
Chemical Name: BMS-P5 free base
Synonyms: BMS-P5; BM P5; BMSP5; BMSP-5; BMSP 5; BMS-P5 HCl; BMS-P5
SMILES: O=C(N1[C@@H](C)CC[C@@H](N)C1)C2=CC(OC)=C3C(N=C(C4=CC5=CC=CN=C5N4CC6CC6)N3C)=C2
Formula: C27H32N6O2
M.Wt: 472.593
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: Li M, Lin C, Deng H, Strnad J, Bernabei L, Vogl DT, Burke JJ, Nefedova Y. A Novel Peptidylarginine Deiminase 4 (PAD4) Inhibitor BMS-P5 Blocks Formation of Neutrophil Extracellular Traps and Delays Progression of Multiple Myeloma. Mol Cancer Ther. 2020 Jul
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