ARQ-087·2HCl|cas 1821329-75-2|DC Chemicals

Cas No.:	1821329-75-2
Chemical Name:	Derazantinib dihydrochloride
Synonyms:	ARQ-087·2HCl;Derazantinib dihydrochloride;Derazantinib hydrochloride;ARQ 087.2HCl;U6B7J0L31Q;AQ14741087;(R)-6-(2-fluorophenyl)-N-(3-(2-((2-methoxyethyl)amino)ethyl)phenyl)-5,6-dihydrobenzo[h]quinazolin-2-amine dihydrochloride;Derazantinib hydrochloride (USAN);Derazantinib hydrochloride [USAN];Derazantinib dihydrochlororide;AMY16761;D11461;Benzo(H)qui
SMILES:	Cl.Cl.FC1C=CC=CC=1[C@H]1C2C=CC=CC=2C2C(=CN=C(NC3=CC=CC(=C3)CCNCCOC)N=2)C1
Formula:	C₂₉H₃₁Cl₂FN₄O
M.Wt:	541.490
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

Derazantinib is a multi-kinase inhibitor with pan-FGFR activity which has shown preliminary therapeutic activity against FGFR2 fusion-positive intrahepatic cholangiocarcinoma (iCCA). Derazantinib dihydrochloride is a salt of Derazantinib.

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2018-0101

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