GN13|cas |DC Chemicals

Cas No.:
Chemical Name:	GN13
Synonyms:	GN 13；GN-13
SMILES:	CC[C@H](C)[C@@H]1NC(=O)[C@H](C)NC(=O)[C@H](CC2=CC=C(O)C=C2)NC(=O)C(C(C)C)NC(=O)[C@H](CO)NC(=O)[C@H](CCC(=O)O)NC(=O)[C@H](CC2=CC=CC=C2)NC(=O)[C@@H](CC2=CC=C(O)C=C2)NC(=O)CSC[C@@H](C(=O)NCC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@H]([C@@H](C)O)NC(=O)CNC(=O)[C@H](CC2=CNC3=C2C=CC=C3)NC1=O
Formula:	C₇₉H₁₀₆O₂₁N₁₆S
M.Wt:	1647.87
Purity:	>98%
Sotrage:	2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO

Description:

GN13 is a cell-permeable, nucleotide-active-state-selective inhibitor of Gαs, with high selectivity over other G protein subfamilies. GN13 binds to Gαs/GNP with KD of 0.19 μM.

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