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GS-4361(IDO-IN-13)

  Cat. No.:  DC30008   Featured
Chemical Structure
2291164-02-6
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More than 5000 active chemicals with high quality for research!
Field of application
GS-4361 is a potent and selective IDO1 inhibitor with an EC50 of 17 nM, GS-4361 was first reported in patent WO2019040102A.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2291164-02-6
Chemical Name: 5-[3-(2,3-Difluorophenyl)imidazo[1,5-a]pyridin-8-yl]-N-(4-fluorophenyl)-2-methyl-3-pyridinecarboxamide
Synonyms: GS-4361; GS 4361; GS4361
SMILES: O=C(NC1C=CC(F)=CC=1)C1C(C)=NC=C(C2C3=CN=C(C4C(F)=C(F)C=CC=4)N3C=CC=2)C=1
Formula: C26H17F3N4O
M.Wt: 458.43
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: GS-4361(IDO-IN-13) is a potent indoleamine 2,3-dioxygenase 1 (IDO1) inhibitor with an EC50 of 17 nM, extracted from patent WO2019040102A1, example 43[1].
Target: EC50: 17 nM[1]
References: [1]. Mark J. BARTLETT, et al. Therapeutic heterocyclic compounds. WO2019040102A1.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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