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IPN-60090 dihydrochloride

  Cat. No.:  DC39259  
Chemical Structure
2102101-72-2
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More than 5000 active chemicals with high quality for research!
Field of application
IPN-60090 dihydrochloride is an orally bioavailable and selective inhibitor of GLS1 (the kidney-type glutaminase), an important enzyme for metabolic energy production. IPN-60090 dihydrochloride can be used in the research of GLS1-mediated diseases[1][2].
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 2102101-72-2
Synonyms: IPN-60090;IPN 60090;IPN60090
SMILES: O=C(C1N=NN(C[C@@H](CCC2C=CC(NC(=O)CC3C=C(OC4CC(F)(F)C4)C=C(C)N=3)=NN=2)F)C=1)NC.[H]Cl.[H]Cl
Formula: C24H29Cl2F3N8O3
M.Wt: 605.44
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Publication: [1]. Maria Emilia Di Francesco, et al. Gls1 inhibitors for treating disease. WO2016004404A2. [2]. Philip Jones, et al. Salt forms and polymorphs of (r)-1-(4-(6-(2-(4-(3,3-difluorocyclobutoxy)-6-methylpyridin-2-yl)acetamido) pyridazin-3-yl)-2-fluorobutyl)-n-methyl-1h-1,2,3-triazole-4-carboxamide. US20170174661A1.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
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