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VL-285

  Cat. No.:  DC12676   Featured
Chemical Structure
1448188-57-5
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More than 5000 active chemicals with high quality for research!
Field of application
VL285 is a potent VHL ligand, degrading HaloTag7 fusion proteins.
Chemicals PropertiesBiological activity COA & MSDSRelated productsDatasheet
Cas No.: 1448188-57-5
Synonyms: VL-285; VL 285; VL285
SMILES: O=C([C@H]1N(C([C@@H](N(CC2=C3C=CC=C2)C3=O)C(C)C)=O)C[C@H](O)C1)NCC4=CC=C(C5=C(C)N=CS5)C=C4
Formula: C29H32N4O4S
M.Wt: 532.66
Purity: >98%
Sotrage: 2 years -20°C Powder, 2 weeks 4°C in DMSO, 6 months -80°C in DMSO
Description: VL285 is a potent VHL ligand.
Target: VHL[1]
References: [1]. Buckley DL, et al. HaloPROTACS: Use of Small Molecule PROTACs to Induce Degradation of HaloTag Fusion Proteins. ACS Chem Biol. 2015 Aug 21;10(8):1831-7.
MSDS
COA
LOT NO. DOWNLOAD
2018-0101
2018-0101
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