Alternate TextTo enhance service speed and avoid tariff delays, we've opened a US warehouse. All US orders ship directly from our US facility.
Home > Products > Novel inhibitors

Novel inhibitors

You can also try the following methods, and our professionals will serve you Customized Consultation
Cat. No. Product Name Field of Application Chemical Structure
DC36330 NSC 33700
γ-Valerolactone is a prodrug form of γ-hydroxyvaleric acid.
More description
DC36294 6(5H)-Phenanthridinone
6(5H)-Phenanthridinone is an inhibitor of poly(ADP-ribose) polymerase 1 (PARP1) and PARP2. It decreases radiation-induced PARP activity and proliferation of RDM4 murine lymphoma cells. 6(5H)-Phenanthridinone reduces NF-κB-induced transcription of the genes encoding TNF-α, IL-2, and IFN-γ in rat lymphocytes. In vivo, 6(5H)-phenanthridinone reduces spinal cord expression of inducible nitric oxide synthase (iNOS), IL-1β, TNF-α, IL-2, and IFN-γ and reduces disease score in a rat model of experimental autoimmune encephalomyelitis (EAE). It also decreases serum levels of lactate dehydrogenase as well as hepatic lipid peroxidation, oxidative DNA damage, and PARP levels.
More description
DC36286 Dihydrocaffeic acid
Dihydrocaffeic acid is a polyphenol with antioxidant, neuroprotective, and enzyme inhibitory properties. Dihydrocaffeic acid scavenges ABTS and 2,2-diphenyl-1-picrylhydrazyl (DPPH) radicals and increases the survival of RGC-5 mouse retinal ganglion cells under hypoxic conditions and in the presence of S-nitroso-N-acetyl-D,L-penicillamine (SNAP). It also decreases endothelial nitric oxide synthase (eNOS) activity and decreases infarct size in a rat model of transient ischemia induced by middle cerebral artery occlusion (MCAO).
More description
DC36210 Amigal
Migalastat is a potent inhibitor of glycolipid biosynthesis.
More description
DC36199 (+)-Amlodipine
(R)-Amlodipine is the R isomer of Amlodipine --- a medication used to lower blood pressure and prevent chest pain.
More description
DC36163 AI3-52333
Gibbs reagent is a universal thin-layer chromatographic visualization reagent.
More description
DC36147 Triphenyltetrazolium bromide
Triphenyltetrazolium bromide may be useful in the detection of experimental cerebral infarction and biochemical analysis.
More description
DC36134 Thioperamide
Thioperamide is an HRH4 antagonist and selective HRH3 antagonist capable of crossing the blood–brain barrier. Thioperamide negatively regulates the release of histamine and enhances the activity of histaminergic neurons by blocking autoreceptors. Its action on H3 is thought to promote wakefulness and improve memory consolidation.
More description
DC36116 AG-1777
Lansoprazole sulfide is an impurity of Lansoprazole -- a gastric pump inhibitor.
More description
DC36110 IMS2186
IMS2186 is an anti-proliferative and anti-angiogenic agent. IMS2186 blocks the cell cycle at G2 and inhibits the production of PGE2/TNF-α. IMS2186 inhibits cell growth in vitro in tumor cells, non-transformed fibroblasts, and retinal pigment epithelial cells. IMS2186 inhibits angiogenesis (IC50 = 0.1 μM) and cell migration. Intraocular injection of IMS2186 could be a long-lasting effective treatment for CNV (choroidal neovascularization) in AMD (age-related macular degeneration) with a reduction in scarring and related visual loss.
More description
DC36102 Aciclovir EP Impurity F
N2-Acetylaciclovir, also known as Aciclovir EP Impurity F, is an impurity of Aciclovir.
More description
DC36056 Aminoform
Methenamine is an anti-infective agent most commonly used in the treatment of urinary tract infections. Its anti-infective action derives from the slow release of formaldehyde by hydrolysis at acidic pH.
More description
DC35960 Ms-PEG8-Ms
Ms-PEG8-Ms is a PEG Linker.
More description
DC35926 PEG5-bis(phosphonic acid diethyl ester)
PEG5-bis(phosphonic acid diethyl ester) is a PEG Linker.
More description
DC35921 Propargyl-PEG3-phosphonic acid ethyl ester
Propargyl-PEG3-phosphonic acid ethyl ester is a PEG Linker.
More description
DC35873 m-PEG5-succinimidyl carbonate
m-PEG5-succinimidyl carbonate is a PEG Linker.
More description
DC35848 Bis-Mal-PEG3
Bis-Mal-PEG3 is a PEG derivative containing a two maleimide groups. The maleimide groups will react with a thiol group to form a covalent bond, enabling the connection of biomolecule with a thiol. The hydrophilic PEG spacer increases solubility in aqueous media.
More description
DC35700 Azido-PEG3-CH2CO2-NHS
Azido-PEG3-CH2CO2-NHS is a PEG Linker.
More description
DC35680 Ald-CH2-PEG3-azide
Ald-CH2-PEG3-azide is a crosslinker containing an azide group and an aldehyde group. The azide group enables PEGylation via Click Chemistry. The hydrophilic PEG spacer increases solubility in aqueous media. The aldehyde group reacts with amines and the N-terminal of peptides and proteins to form an imine containing a C=N double bond, which can be further reduced. PEG aldehyde or ketone derivatives can be used in reversible PEGylation through its reaction with hydrazine or hydrazide forming a hydrolytic acyl hydrozone linkage.
More description
DC35629 Sulfo-NHS
Sulfo-NHS is a chemical modification reagent for converting carboxyl groups to amine-reactive NHS esters for bioconjugation, crosslinking, labeling and immobilization methods.
More description
DC35617 diethyl 7-bromoheptylphosphonate
diethyl 7-bromoheptylphosphonate is a PEG Linker.
More description
DC35589 m-PEG3-4-nitrophenyl carbonate
m-PEG3-4-nitrophenyl carbonate is a PEG derivative.
More description
DC35579 m-PEG13-Ms
m-PEG13-Ms is a PEG Linker
More description
DC35569 m-PEG4-CH2-aldehyde
m-PEG4-CH2-aldehyde is a PEG derivative containing an aldehyde group. Aldehyde is reactive to hydrazide and aminooxy groups which are commonly used in biomolecular probes for labeling and crosslinking carbonyls (oxidized carbohydrates). The hydrophilic PEG spacer increases solubility in aqueous media.
More description
DC35556 m-PEG6-azide
m-PEG6-azide is a PEG derivative containing an azide group. The azide group can react with alkyne, BCN, DBCO via Click Chemistry to yield a stable triazole linkage. The hydrophilic PEG spacer increases solubility in aqueous media.
More description
DC35533 m-PEG1-NHS ester
m-PEG1-NHS ester is a PEG derivative containing an NHS ester. The NHS ester can be used to label the primary amines (-NH2) of proteins, amine-modified oligonucleotides, and other amine-containing molecules. The hydrophilic PEG spacer increases solubility in aqueous media.
More description
DC35531 m-PEG9-CH2COOH
m-PEG9-CH2COOH is a PEG derivative containing a terminal carboxylic acid. The terminal carboxylic acid can be reacted with primary amine groups in the presence of activators (e.g. EDC, or DCC) to form a stable amide bond. The hydrophilic PEG spacer increases solubility in aqueous media.
More description
DC35512 Tri(t-butoxycarbonylethoxymethyl) ethanol
Tri(t-butoxycarbonylethoxymethyl) ethanol is a branched PEG derivative with a terminal hydroxy group and three t-butyl esters. The hydroxy group enables further derivatization or replacement with other reactive functional groups. The t-butyl protected carboxyl groups can be deprotected under mild acidic conditions.
More description
DC35477 Tr-PEG3
Tr-PEG3 is a PEG derivative.
More description
DC35466 m-PEG3-(CH2)3-alcohol
m-PEG3-(CH2)3-alcohol is a PEG derivative containing a hydroxyl group. The hydroxyl group enables further derivatization or replacement with other reactive functional groups. The hydrophilic PEG spacer increases solubility in aqueous media.
More description

Customized Consultation X

Your information is safe with us. * Required Fields.

Your name
Company
Email
Procuct Name
Cat. No.
Remark
Verification code
Please fill out the characters in the picture
X