Cheirolin is an antioxidant and sulfonyl analog of sulforaphane. It induces phase II enzyme activity and expression.

Ceftiofur sodium is a penicillin binding protein inhibitor that prevents synthesis of bacterial cell walls. It also decreases LPS-induced expression of pro-inflammatory cytokines in endotoxemia models.

Cefotaxime Acid is a penicillin binding protein inhibitor that prevents peptidoglycan synthesis and bacterial cell wall formation. It is mostly resistant to β-lactamase activity.

Cefoperazone is a penicillin binding protein inhibitor and mammalian mRNA splicing inhibitor that prevents peptidoglycan synthesis and bacterial cell wall formation.

Cefaclor monohydrate is a penicillin binding protein inhibitor that prevents peptidoglycan synthesis and bacterial cell wall formation. It also enhances phagocytosis, bacterial activity of granulocytes and macrophages, and slows gastric emptying and intestinal transit.

Canrenone is a metabolite of spironolactone, Na/K ATPase partial agonist and aldosterone and androgen receptor antagonist used as a diuretic.

Cerulomycin A is a toxin that inhibits growth of Entamoeba. It may prevent proliferation of cancer cells, and suppresses immune responses.

Butein is found in Rhuteic verniciflua and Butea monosperma. It induces cell cycle arrest and apoptosis in lung cancer cells, inhibits vessel spouting from aortic rings, and prevents hepatic stellate cell activation.

Bupivacaine is a BK/SK, Kv1, Kv3, TASK-2 K Channel and voltage-gated Na channel blocker used as an anesthetic. It maybe neurotoxic at high does, inducing apoptosis in neuroblastoma cells.

Biopterin is an endogenous pterin coenzyme required for production of neutrotransmitters and release of NO

Ubenimex, also known as NK 421 and Bestatin, is a CD13 inhibitor. Ubenimex attenuates acquired sorafenib resistance in renal cell carcinoma by inhibiting Akt signaling in a lipophagy associated mechanism. Ubenimex synergistically enhances the effects of anticancer drugs in hepatocellular carcinoma. Ubenimex inhibits cell proliferation, migration and invasion by inhibiting the expression of APN and inducing autophagic cell death in prostate cancer cells.

Berteroin is an erucin homolog and potential antioxidant. It is present in cruciferous vegetables, including Chinese cabbage, rucola salad leaves, and mustard oil. It decreases expression of androgen receptors in prostate cancer cells. It also decreases the release of pro-inflammatory cytokines in LPS-stimulated macrophages.

Azithromycin dihydrate is a protein translation inhibitor used for it's antibacterial properties. It is also known to inhibit the epithelila-to-mesenchymal transition and suppresses LPS-stimulated production of pro-inflammatory cytokines in macrophages.

Atropine is a mAChR antagonist found in Solanaceae used to initiate mydriasis. It decreases thermal pain, inhibits histamine-induced increases in thromboxane A2, and acts as a positive inotrope.

Antipain HCl is a protease inhibitor found in Actinomycetes.

Anisodamine is an inhibitor of alpha-1 adrenergic receptors and mAChRs isolated from Chinese solanacea plant.

Anabasine HCl is used as an insecticide and as a clinical biomarker for tobacco smoke exposure. It is also a depolarizing NMJ blocker, nAChr antagonist, aromatase inhibitor, and teratogen found in species of Nicotiana.

Amprolium HCl is coccidiostat and thiamine transporter inhibitor. It inhibits thiamine transporters in species of Eimera, preventing carbohydrate synthesis.

Ampicillin Trihydrate is a transpeptidase inhibitor that prevents bacterial cell wall formation. It is effective against gram negative and gram positive bacteria.

Amitraz, also known as Mitaban and Taktic, is an alpha-adrenergic receptor agonist and MAO inhibitor used as an insecticide in prevention of flea and tick infections. It prevents prostaglandin synthesis and may inhibit beta-cell insulin release.

Amisulpride is an antagonist 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.

Alyssin is a sulforaphane homolog and antioxidant. It induces phase II enzymes and increases Nrf2 levels in adenocarcinoma cells. It is has been shown to decrease the metabolism of polycyclic aromatic hydrocarbons, supressing the risk of carcinogenesis in vitro.

Alternariol is a mycotoxin, topoisomerase I and II inhibitor and potential ER agonist found in Alternaria.

Acepromazine maleate, also known as Sch-10649, is a dopamine D1/2 receptor and 5-HT1A/2A receptor antagonist used to prevent nausea and induce sedation. Acepromazine maleate is discontinued.

Pramiverin HCl is a bioactive chemical.

MS4 is a novel glucocorticoid receptor (GR) agonist with anti-inflammatory activity and displaying reduced impact on islets.

Nevirapine-d3 is deuterized nevirapine, reducing P450 metabolite formation, impacting on phase II metabolism and hepatocyte protein expression.

Garcinoic Acid is a natural and selective agonist of pregnane X receptor.

Levothyroxine sodium is a thyroid hormone.

Oxacillin (trade name Bactocill) is a narrow-spectrum beta-lactam antibiotic of the penicillin class developed by Beecham. It was patented in 1960 and approved for medical use in 1962. Oxacillin is a penicillinase-resistant β-lactam. It is similar to methicillin, and has replaced methicillin in clinical use.