Procaterol is an intermediate-acting β2 adrenoreceptor agonist used for the treatment of asthma.

H2DCFDA is a fluorescent cell permeabl ROS indicator.

PNU-142633 selective, high affinity 5-HT1D receptor antagonist and is an experimental drug candidate for the treatment of migraine.

Fenpyroximate is an acaricide and insecticide, blocking the mitochondrial electron transport in complex I.

rac-CCT-250863 is a potent Nek2 inhibitor. exhibiting selectivity for Nek2 over PLK1, MPS1, Cdk2 and Aurora A.

HHQ is an antagonist of PqsR.

Sulfaclozine is an antiprotozoal.

Piromidic acid is antibacterial against mainly gram negative organisms. It is used for urinary tract and intestinal infections.

Physostigmine salicylate is a reversible cholinesterase inhibitor, a parasympathomimetic alkaloid. It also can cross the blood-brain barrier and is used when central nervous system effects are desired, as in the treatment of severe anticholinergic toxicity.

PDP-EA is an FAAH activator, enhancing amidohydrolase activity of FAAH.

Levoglucosenone is a cytotoxic, against human hepatocarcinoma cell lines.

PBI-51 is a competitive Inhibitor of Abscisic Acid-Regulated Gene Expression.

Propachlor is a specific ALDH1A1 inhibitor. It is sometimes used as an herbicide.

L-670596 is a potent and selective thromboxane A2/prostaglandin endoperoxide receptor antagonist, also showing ALDH1A1 specific inhibitory activity.

Desmosterol is an endogenous agonist of RORgamma; Intermediate in the synthesis of cholesterol.

Rauwolscine hydrochloride is an alpha2-Adrenergic antagonist and partial agonist at 5-HT1A receptors.

Sulfidefluor-7 AM is a novel hydrogen sulphide (H2S) fluorescent probe.

Fenirofibrate is a metabolite of Fenofibrate.

LP117 is a novel drug-specific modulator of ABCB1-mediated drug transport.

Periciazine is a drug that belongs to the phenothiazine class of typical antipsychotics. Periciazine is used to treat short-term severe anxiety or tension and in the maintenance treatment of psychotic disorders such as schizophrenia.

Pencycuron, also known as Monceren, is a phenylurea fungicide.

PD-198306 is a cell-permeable amino-benzamide compound that acts as a potent and non-ATP-competitive inhibitor of MEK1/2 (IC50 = 8 nM) with an excellent selectivity over ERK, c-Src, Cdk's, and PI 3-Kγ (IC50 >1.0 μM).

NCL00017509 is a potent and reversible NIMA related kinase 2 (Nek2) inhibitor.

PD-176252 is a non-peptide gastrin-releasing peptide receptor (GRP-R, BB2) and neuromedin B receptor (NMB-R, BB1) antagonist (Ki values are 0.17 and 1.0 nM for BB1 and BB2 respectively). It inhibits proliferation of rat C6 glioma cells (IC50 = 2 μM) and inhibits NCI-H1299 xenograft proliferation in nude mice (IC50 = 5 μM).

TrxR-IN-D9, also known as D9, is a novel inhibitor of thioredoxin reductase (TrxR).

Tiaprost is a prostaglandin F2 alpha analogue as an estrus-synchronizing agent.

NB-64 is a novel human immunodeficiency virus type 1 (HIV-1) entry inhibitor, interferring with the gp41 six-helix bundle formation and blocking virus fusion.

Nitrocefin is an antibiotic, being sensitive to hydrolysis by all lactamases produced by gram-positive and gram-negative bacteria.

Oxantel is a fumarate reductase inhibitor; Anthelmintic.

(S)-alpha-Fluoromethylhistidine HCl is a potent irreversible histidine decarboxylase (HDC) inhibitor and glutathione S-transferase inhibitor. a-FMH was demonstrated to be an effective inhibitor of GST at micromolar concentration, suggesting that off-target effects of a-FMH may limit physiological drug metabolism and elimination by GST-dependent mechanisms.