To enhance service speed and avoid tariff delays, we've opened a US warehouse. All US orders ship directly from our US facility.
| Cat. No. | Product Name | Field of Application | Chemical Structure |
|---|---|---|---|
| DC12517 | HT105 |
DB550 (DB-550, TCWKHRK) is a potent, peptidomimetic of calcium-inducing domain (CID) that disrupts the CD95-PLCγ1 interaction, abrogates the CD95-mediated Ca2+ response in mouse PBLs with IC50 of 38 nM.
More description
|
|
| DC12516 | DB550 |
DB550 (DB-550) is a potent, peptidomimetic of calcium-inducing domain (CID) that disrupts the CD95-PLCγ1 interaction without affecting the CD95-FADD interaction binds to SH3-PLCγ1 with Kd of 40.7 uM.
More description
|
|
| DC20943 | DB2115 |
DB2115 is a small-molecule transcription factor PU.1 inhibitor abrogating DNA binding by PU.1 with Kd of 1.0 nM.
More description
|
|
| DC22067 | DB1055 |
DB1055 (DB-1055, DB 1055) is a small molecule inhibitor of HOXA9/DNA interaction through binding as minor groove DNA ligand on the HOXA9 cognate sequence.
More description
|
|
| DC20942 | DB04760 |
DB04760 is a potent, highly selective, non–zinc-chelating MMP-13 inhibitor with IC50 of 8 nM, displays high selectivity over other MMPs.
More description
|
|
| DC9331 | Daun02 |
Daun02 is a daunorubicin b-galactoside prodrug for use in conjunction.
More description
|
|
| DC21381 | Dasolampanel |
Dasolampanel (NGX426) is an orally bioavailable, competitive antagonist of the AMPA-kainate receptors for the treatment of chronic pain conditions including neuropathic pain and migraine..
More description
|
|
| DC2100 | Dasatinib (BMS-354825) Featured |
Dasatinib (BMS-354825, Sprycel) is a novel, potent and multi-targeted inhibitor that targets Abl, Src and c-Kit, with IC50 of <1 nM, 0.5 nM and 79 nM, respectively.
More description
|
|
| DC3152 | Darifenacin |
Darifenacin is a selective M3 muscarinic receptor antagonist with pKi of 8.9.
More description
|
|
| DCAPI1440 | Darifenacin HBr |
Darifenacin Hydrobromide is an antagonist of the M3 musarinnic acetylcholine receptor.
More description
|
|
| DC10259 | Dapson |
Dapsone, also known as diaminodiphenyl sulfone (DDS), is an antibiotic commonly used in combination with rifampicin and clofazimine for the treatment of leprosy.
More description
|
|
| DC20354 | DAPH-12 |
DAPH-12 is a small molecule that directly inhibits and reverses prion protein Sup35 prionogenesis (IC50=0.18 uM).
More description
|
|
| DC9116 | Dantrolene sodium |
Dantrolene sodium is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ from the sarcoplasm. Dantrolene sodium is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction.
More description
|
|
| DC8665 | Dantrolene sodium hemiheptahydrate |
Dantrolene sodium hemiheptahydrate is a skeletal muscle relaxant which acts by blocking muscle contraction beyond the neuromuscular junction. Dantrolene sodium hemiheptahydrate is a inhibitor of calcium channel proteins, inhibiting the release of Ca2+ fro
More description
|
|
| DC12338 | Dansylamide |
Dansyl amide is a fluorescent dye that is used in biochemistry and chemistry to label substances with the fluorescent dansyl group.
More description
|
|
| DCAPI1028 | Danofloxacin Mesylate |
Danofloxacin Mesylate
More description
|
|
| DC22810 | Damnacanthal |
Damnacanthal is a highly potent, selective inhibitor of p56 lck tyrosine kinase with IC50 of 17 nM for inhibition of p56lck autophosphorylation.
More description
|
|
| DC21469 | Dagrocorat |
Dagrocorat (PF 00251802) is a potent, selective high-affinity dissociated agonist of the glucocorticoid receptor..
More description
|
|
| DC11232 | D715-2441 |
D715-2441 (D 715-2441) is a novel antiviral compound that interferes with the conserved cap-binding domain of the PB2 protein, exhibits potent antiviral activity against influenza A viruses (IAVs) with IC50 of 1.7-4.4 uM.
More description
|
|
| DC11124 | D-520 |
D-520 is a potent, multifunctional D2/D3 agonist with Ki of 41.8 /0.35 nM, modulates aggregation of alpha-synuclein (αSN) and reduces toxicity of preformed aggregates of αSN.
More description
|
|
| DC12610 | D159153 |
D159153 (D-159153) is a novel potent, allosteric inhibitor of PDE4 with cellular IC50 of 28.5 and 6.6 nM for PDE4B1 and PDE4D3, respectively..
More description
|
|
| DC25001 | D-156844 |
D156844 is a potent SMN2 inducer and DcpS inhibitor.
More description
|
|
| DC12582 | D13-9001 |
D13-9001 (D 13-9001) is a small molecule, MexAB-OprM specific efflux pump inhibitor with good potency in vitro (MPC 2 ug/mL) and displays excellent activity in vivo in a rat pneumonia model of P. aeruginosa..
More description
|
|
| DC9886 | D-(+)-Cellobiose |
D-(+)-Cellobiose is a substrate of β-glucosidase.
More description
|
|
| DC11198 | CZh226 hydrochloride |
CZh226 hydrochloride (CZh-226) is a potent, selective inhibitor of p21-activated kinase 4 (PAK4) with Ki of 9 nM, displays 346-fold selectivity over PAK-1.
More description
|
|
| DC5134 | lexibulin (CYT997) |
CYT997 is a potent microtubule polymerization inhibitor with IC50 of 10-100 nM in cancer cell lines. Phase 1/2.
More description
|
|
| DCAPI1536 | Cyproheptadine Hydrochloride |
Cyproheptadine hydrochloride is a migraine prophylactic and Non-selective SR-2A (5HT2) antagonist. Cyproheptadine hydrochloride is an inhibitor of Histamine H1 Receptor and SR-2C.
More description
|
|
| DC20352 | CYP11B1-IN-25 |
CYP11B1-IN-25 is a selective, potent 11β-hydroxylase (CYP11B1) inhibitor with IC50 of 2 nM, displays 14-fold selectivity over CYP11B2.
More description
|
|
| DC12470 | CYH33 methanesulfonate |
CYH33 (CYH-33) is a novel potent, PI3Kα-selective inhibitor with IC50 of 5.9 nM/598 nM/ 78.7 nM/225 nM aginst class I PI3K isoform α/β/δ/γ, respectively.
More description
|
|
| DC23283 | CYD-2-11 |
CYD-2-11 is a novel potent, selective Bax agonist that targets the structural pocket proximal to S184 in the C-terminal region of Bax (Ki=34.1 nM).
More description
|
|