XR8-69 is a SARS-CoV-2 PLpro inhibitor that shows low micromolar antiviral potency in SARS-CoV-2-infected human cells.

Undecane has anti-allergic and anti-inflammatory activities on sensitized rat basophilic leukemia (RBL-2H3) mast cells and HaCaT keratinocytes. In sensitized mast cells, Undecane inhibits degranulation and the secretion of histamine and TNF-α.

Palmaturbine hydroxide is isolated from T. sinensis.

Phytohemagglutinin P (PHA-P) is a mitogen known to selectively stimulate cells of hematogenous or lymphoid monocytic origin.

Streptokinase is a bacteria-derived protein and a plasminogen activator. Streptokinase is widely used for the research of the blood-clotting disorders. Streptokinase improves reperfusion blood flow after coronary artery occlusion.

P8RI (D-P8RI) is a biomimetic peptide of CD31 and a CD31 agonist. P8RI binds to the juxtamembrane amino acid sequence of the ectodomain of CD31, shows an immunosuppressive effect through restoration of the CD31 inhibitory pathway.

Micromonosporamide A exhibits glutamine-dependent antiproliferative activity.

NBD-LLLLpY is an enzymatically forming intranuclear peptide for selectively killing human induced pluripotent stem cells.

Pinofuranoxin A completely inhibits the growth of Athelia rolfsii and Phytophthora cambivora.

Penispidin A inhibits hepatic lipid accumulation in HepG2 cells.

Stipuleanoside R2 inhibits NF-κB activation stimulated by TNFα in a dose-dependent manner with IC50 value of 4.1 μM.

Neonuezhenide exhibits strong antioxidant effect against hemolysis of red blood cells induced by free radicals.

Scutebarbatine B shows significant cytotoxic activities against three human cancer lines, namely, HONE-1 nasopharyngeal, KB oral epidermoid carcinoma, and HT29 colorectal carcinoma cells, with IC50 values in the range 3.5-8.1 mM.

Odoratisol A is found in Myristica fragrans.

L-Borneol 7-O-[β-D-apiofuranosyl-(1→6)]-β-D-glucopyranoside is one of the components of the Shengmai injection.

Ruscogenin suppresses HCC metastasis by reducing the expression of MMP-2, MMP-9, uPA, VEGF and HIF-1α via regulating the PI3K/Akt/mTOR signaling pathway. And Ruscogenin alleviates LPS-induced pulmonary endothelial cell apoptosis by su

Sanggenone H is found in Morus alba L.

Oleoside 11-methyl ester is a secoiridoid glucoside and possesses a strong cytotoxic activity against Hep-G2 cells.

Methyl p-hydroxyphenyllactate (MeHPLA) is an important cell growth-regulating agent which binds to nuclear type II binding sites in normal and malignant cells.

Pinosylvin monomethyl ether has antibacterial effect and fungicidal activity.

Kulinone has cytotoxic effects against A549, H460 and HGC27 with IC50 values of 6.2 ± 0.1, 7.8 ± 1.2, 5.6 ± 0.2 μg/ml。

Samwirin A is a promising radical scavenger in aqueous media at physiological pH.

Suomilide inhibits human trypsin-2 and -3, with IC50 values of 4.7 and 11.5 nM, respectively, while trypsin-1 is inhibited with an IC50 of 104 nM.

Rhodiocyanoside A is found to show antiallergic activity in a passive cutaneous anaphylaxis test in rat.

Rocaglaol induces apoptosis and cell cycle arrest in LNCaP cells.

Rotundatin is useful in inhibition of the aggregation of platelets induced by arachidonic acid and collagen.

Monnieriside G is found in Cnidium monnieri fruits.

Methylsyringin exhibits anti-inflammatory activity in the LPS-stimulated RAW264.7 cells.

Rutaretin is found in Atalantia racemosa.

Quebecol is a nutraceutical agent against periodontitis.