Antagonist of the actions of ethanol, attenuating the ethanol-induced reduction in cerebellar cyclic guanosine monophosphate (cGMP) content, but significantly elevating cGMP levels when given alone

Novel highly potent, selective, and irreversible GSTP1 inhibitor

Prodrug of Fenclonine as a selective and irreversible inhibitor of tryptophan hydroxylase

NMDA antagonist acting at the polyamine site; Neuroprotective agent; α-Adrenergic central and peripheral vasodilator; α2 adrenergic receptor ligand

Used experimentally as a beta blocker and clinically as a strong vasodilator with the noted side effects of reduced systolic, diastolic and mean arterial pressure.

Yoda1 analogue, antagonizing Yoda1-evoked activation of Piezo1 and aortic relaxation.

Novel subtilisin kexin isozyme-1/site-1 (SKI-1/S1P) protease inhibitor