Sanggenone H is found in Morus alba L.

Oleoside 11-methyl ester is a secoiridoid glucoside and possesses a strong cytotoxic activity against Hep-G2 cells.

Methyl p-hydroxyphenyllactate (MeHPLA) is an important cell growth-regulating agent which binds to nuclear type II binding sites in normal and malignant cells.

Pinosylvin monomethyl ether has antibacterial effect and fungicidal activity.

Kulinone has cytotoxic effects against A549, H460 and HGC27 with IC50 values of 6.2 ± 0.1, 7.8 ± 1.2, 5.6 ± 0.2 μg/ml。

Samwirin A is a promising radical scavenger in aqueous media at physiological pH.

Suomilide inhibits human trypsin-2 and -3, with IC50 values of 4.7 and 11.5 nM, respectively, while trypsin-1 is inhibited with an IC50 of 104 nM.

Rhodiocyanoside A is found to show antiallergic activity in a passive cutaneous anaphylaxis test in rat.

Rocaglaol induces apoptosis and cell cycle arrest in LNCaP cells.

Rotundatin is useful in inhibition of the aggregation of platelets induced by arachidonic acid and collagen.

Monnieriside G is found in Cnidium monnieri fruits.

Methylsyringin exhibits anti-inflammatory activity in the LPS-stimulated RAW264.7 cells.

Rutaretin is found in Atalantia racemosa.

Quebecol is a nutraceutical agent against periodontitis.

Peucedanocoumarin II can induce rice resistance to blast disease.

OJV-VI is found in ophiopogonis.

Schisanwilsonin B is a lignan from the fruits of Schisandra wilsoniana.

Moscatin inhibits AA-induced platelet aggregation in a concentration-dependent manner with IC50 values 37.2 μM .

Olivil monoacetate is found in Gymnosporia varialilis Loes.

Mulberrofuran Q inhibits the formation of 12-hydroxy-5,8,10-heptadecatrienoic acid (HHT) and thromboxane B2 (cyclooxygenase products).

Nurr1 agonist 1 is an inverse agonist tool for the neuroprotective transcription factor Nurr1.

Oxythiamin diphosphate ammonium is a potent transketolase (TK) inhibitor.

SLK/STK10-IN-1 is a potent and selective inhibitor of SLK and STK10 with nanomolar potency.

SPOP-IN-6b dihydrochloride is a potent speckle-type POZ protein (SPOP) inhibitor with an IC50 of 3.58 μM.

Sinbaglustat (OGT2378) is a dual inhibitor of glucosylceramide synthase (GCS) and non-lysosomal glucosyl ceramidase (GBA2). Sinbaglustat is an orally available N-alkyl iminosugar that crosses the blood-brain barrier. Sinbaglustat can be used for the research of central neurodegenerative diseases associated with lysosomal dysfunctions.

R-(+)-Cotinine ((+)-Cotinine), a Nicotine metabolite, lacks significant activity across a wide range of pharmacological targets. R-(+)-Cotinine can enhance the Ach-evoked current in human α7 nAChRs.

Peptide 78, a chemotactic cytokine, a 78 amino acid protein member of the IL-8 or C-X-C chemokine supergene family. ENA-78 plays an important role in the elicitation of predominantly neutrophils (PMNs) into the joints of rheumatoid arthritis (RA).

TIM-3-IN-1 represents useful tool to further study the biology of TIM-3 immune modulation in cancer.

PREP inhibitor-1 is a highly potent prolyl oligopeptidase (PREP) inhibitor (IC50 < 1 nM).

MEIS-IN-3 is a potent myeloid ecotropic viral integration site (MEIS) inhibitor.