CTP354, also known as C-21191, a novel deuterated subtype-selective GABA(A) modulator. CTP may be potentially useful for treatment of neuropathic pain, spasticity and anxiety disorders. GABAA receptors are found in the nervous system and, when activated, reduce the transmission of certain nerve signals. Several classes of widely used drugs target GABAA receptors, including benzodiazepines, but do not have the receptor subtype selectivity of CTP-354.

HPK1-IN-2 is a potent and orally active inhibitor of hematopoietic progenitor kinase-1 (HPK1, a serine/threonine Ste20-related protein kinase), Lck and Flt3 with IC50 of <0.05 μM, IC50 of <0.5 μM and IC50 of <0.05 μM, respectively. HPK1-IN-2 exhibits antitumor activity.

5'-N-Ethylcarboxamidoadenosine (NECA, 5'-(N-Ethylcarboxamido)adenosine, Adenosine-5'N-ethylcarboxamide, 5'-Ethylcarboxamidoadenosine) is a stable, nonselective adenosine receptor agonist. 5'-N-Ethylcarboxamidoadenosine acts via multiple mechanisms including: reducing diabetes-induced oxidative stress, inhibiting gene expression of IL-18, TNF-α and ICAM-1 (intercellular adhesion molecule 1 (CD54)), and blocking activation of the JNK-MAPK pathway.

Protamine sulfate, polycationic peptide and a antiheparin agent, could neutralize the anticoagulant action of heparin and enhances lipid-mediated gene transfer.

POT-4 TFA (AL-78898A TFA), a Compstatin derivative, is a potent inhibitor of complement factor C3 activation. POT-4 TFA can be used for age-related macular degeneration research.

Deltorphin 2 TFA is a selective peptide agonist for the δ opioid receptor.

Stachyose hydrate act as a prebiotic to enhance the growth and activity of beneficial bacteria. Stachyose hydrate exhibit a hypoglycemic effect, and improve inflammation through modulating gut microbiota.

Sodium carboxymethyl cellulose (CMC-Na) (MW 250000) is the sodium salt of cellulose arboxymethyl and frequently used as viscous agent, paste and barrier agent.

Wilfortrine is a bioactive sesquiterpene alkaloid. Wilfortrine exhibits immunosuppresive effects. Wilfortrine also can inhibit leukaemia cell growth in mice and shows anti-HIV activity.

Vindolinine is a natural alkaloide that can be found in Catharanthus roseus.

Tetradehydropodophyllotoxin possesses antifungal activity.

Schisanwilsonin C (Arisanschinin K) shows anti-HBV activity.

Neoisoastilbin possesses antioxidant, anti-hyperuricemic and anti-Inflammatory activities.

Methyl caffeate, an antimicrobial agent, shows moderate antimicrobial and prominent antimycobacterial activities. Methyl caffeate also exhibits α-glucosidase inhibition activity, oxidative stress inhibiting activity, anti-platelet activity, antiproliferative activity in cervix adenocarcinoma and anticancer activity in lung and leukmia cell lines.

Kaempferol-3-O-(2''-O-β-D-glucopyl)-β-D-rutinoside is a natural glycoside that could be found in Camellia oleifera seeds.

Cantleyoside is a natiural iridoid glycoside that could be found in the Roots of Dipsacus asper.

Broussoflavonol F possess xanthine oxidase inhibitory activity.

Brassicin, a natural Flavonoid, possesses radical scavenging activity.

Brandioside is a natural phenylpropanoid glycoside from Brandisia hancei.

Bletilol B is a natural compound that could be found in Bletilla striata.

Bletilloside A is a natural glucoside that could be found in the tubers of Bletilla striata.

Bisabolone oxide A is an α-glucosidase inhibitor.

Bisabolol oxide A possesses antihyperalgesic and antiedematous effects with oral activity.

Bis(dihydrochelerythrinyl)amine possesses anti-bacteria activity.

Bergaptol O-β-D-glucopyranoside possesses anti-gastric ulcer and anti-cancer effect.

Azedarachol possesses antifeedant activity.

Arundinin is a stilbenoid from Bletilla striata.

Argentinogenin is a natural compound with anti-cancer activity that could be found in traditional Chinese drug Chan Su.

Ardisicrenoside A exhibits anti-cancer activity.

Ardisiacrispin B displays cytotoxic effects in multi-factorial drug resistant cancer cells via ferroptotic and apoptotic cell death.