Novel mixed μ opioid receptor (MOR) agonist and δ/κ opioid receptor (DOR/KOR) antagonist

Novel inhibitor of sterol regulatory element-binding protein (SREBP), impairing the SREBP activity by inhibiting glucose transporters and thereby activating AMP-activated protein kinase (AMPK)

Peptide substrate for many protein kinases, such as Blk, BTK, cKit, EPHA1, EPHB2, EPHB3, ERBB4, FAK, Flt3, IGF-1R, ITK, Lck, MET, MUSK, Ret, Src, TIE2, TrkB, VEGF-R1 (Flt-1) and VEGF-R2 (KDR)

Novel Selective TBK1/IKK dual inhibitor with anticancer potency

The first selective β3 adrenergic agonist, showing to possess a profile of antidepressant activity in rodents

Novel renin inhibitor

Novel Inhibitor of c-Jun N-terminal Kinase 3 (JNK3)

Potent inhibitor of both JNK3 and p38

Novel NR4A nuclear receptor modulator

Novel partial agonist of PPARgamma

Novel Unc-51-Like Kinase 1 (ULK1)

Selective neurotensin antagonist

Novel NR4A nuclear receptor modulator

Novel NR4A nuclear receptor modulator

Novel inhibitor of the in vivo aggregation of

Novel specific PAK4 inhibitor, effectively inhibiting the invasion of SGC7901 cells without cytotoxicity, regulating the PAK4/LIMK1/cofilin and PAK4/SCG10 signaling pathways

Novel potent and selective binder of small subunit B of the serine palmitoyltransferase complex (SPTSSB)

Novel potent serine palmitoyl transferase (SPT) inhibitor

Novel SPOP inhibitor, suppressing the viability and inhibiting the colony formation of ccRCC cell lines driven by cytoplasmic SPOP

Pivotal intercellular signal transmitter

USP7 inhibitor from the marine sponge Stylissa massa

Novel isosteric charge-deficient spermine analogue

Novel potent sPLA2 inhibitor, selectively targeting hGIIA and hGIID

Sterol Biosynthesis Inhibitor, Fungicide

Novel p53 Stabilizer for Brain Cell Differentiation

Novel selective orally bioavailable inhibitor of p300/CBP histone acetyltransferase

Novel gamma-secretase modulator

Antibiotic, binding to the bacterial 30S ribosomal subunit, interfering with the initiation of protein synthesis and with proper protein elongation and leading to bacterial cell death

Novel anti-tuberculosis agent against intracellular Mycobacterium tuberculosis

Novel photo-controllable hydrogen sulfide donor applicable in live cells